SYNTHESIS OF QUINOLIN-2-ONES BY AN INTRAMOLECULAR KNOEVENAGEL CONDENSATION AND BY TANDEM MICHAEL-KNOEVENAGEL HETEROCYCLIZATION
DOI:
https://doi.org/10.1007/1394Keywords:
acyl-2-(N-acylamino)benzenes, acyl-2-vinylcarbonylaminobenzenes, quinolin-2-ones, intramolecular Knoevenagel condensation, tandem heterocyclizationAbstract
The synthesis of 2-(N-R-amino)- and 2-(N-vinylcarbonylamino)acylbenzenes has been carried out and their heterocyclization into quinolin-2-ones under the action of sodium ethylate has been studied.
Authors: S. S. Mochalov, M. I. Chasanov, A. N. Fedotov, and N. S. Zefirov.
English translation in Chemistry of Heterocyclic Compounds, 2011, 47 (9), pp 1105-1121