4-HYDROXY-2-QUINOLONES. 40. SYNTHESIS AND BIOLOGICAL PROPERTIES OF ANILIDES OF 1H-2-OXO-4-HYDROXYQUINOLINE-3-CARBOXYLIC ACID

Authors

  • И. B. Украинец National Pharmaceutical Academy of Ukraine, Kharkov
  • C. Г. Таран National Pharmaceutical Academy of Ukraine, Kharkov
  • O. B. Горохова National Pharmaceutical Academy of Ukraine, Kharkov
  • E. А. Таран National Pharmaceutical Academy of Ukraine, Kharkov
  • Нидаль Амин Джарадат National Pharmaceutical Academy of Ukraine, Kharkov
  • И. Ю. Петухова National Pharmaceutical Academy of Ukraine, Kharkov

DOI:

https://doi.org/10.1007/46

Keywords:

anilide, carbostyryl, 4-hydroxy-2-quinolone, antithyroid activity, antituberculotic action

Abstract

An improved method for the synthesis of anilides of 1H-2-oxo-4-hydroxyquinoline-3-carboxylic acid was proposed. Results of the study of antithyroid and anti-tuberculosis activity of the compounds synthesized are presented.

Authors: I. V. Ukrainets, S. G. Taran, O. V. Gorokhova, E. A. Taran, N. A. Jaradat, and I. Yu. Petukhova.

English Translation in Chemistry of Heterocyclic Compounds, 2000, 36 (2), pp 166-169

http://link.springer.com/article/10.1007/BF02283545

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Published

2012-11-16

Issue

No. 2 (2000)

Section

Original Papers