CONDENSATION OF ETHYL 2-OXOINDOLINE-3-GLYOXYLATE WITH <i>o</i>-AMINOPHENOL AND <i>o</i>-PHENYLENEDIAMINE

Authors

  • В. В. Болотов National Pharmaceutical University, Kharkov, 61002
  • С. Н. Коваленко National Pharmaceutical University, Kharkov, 61002
  • С. В. Ковалева National Pharmaceutical University, Kharkov, 61002
  • В. И. Степаненко National Pharmaceutical University, Kharkov, 61002

Keywords:

2H-1,4-benzoxazin-3(4H)-one, 1,4-dihydroquinoxalin-2-one, 2-oxo-1,2-dihydro-1H-indole, cis-trans izomerism

Abstract

A method is presented for the synthesis of 3-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)-1,4-dihydroquinoxalin-2-one and 2-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)-2H-1,4-benzoxazin-3(4H)-one by the reaction of ethyl 2-oxoindoline-2-glyoxylate with o-aminophenol and o-phenylenediamine. Proposed reaction mechanisms are presented.

How to Cite
Bolotov, V. V.; Kovalenko, S. N.; Kovaleva, S. V.; Stepanenko, V. I. Chem. Heterocycl. Compd. 2004, 40, 211. [Khim. Geterotsikl. Soedin. 2004, 249.]

For this article in the English edition, see DOI 10.1023/B:COHC.0000027894.55256.81

Published

2004-02-25

Issue

Section

Original Papers