Synthesis of pyrroloquinolines from alkyl-substituted 6-aminoindoles, acetoacetic ester, and ethoxymethylenemalonic ester

Authors

  • C. А. Ямашкин M. E. Evsev'ev Mordovian State Pedagogical Institute, Saransk 430007
  • Н. Я. Кучеренко M. V. Lomonosov Moscow State University, Moscow 119899
  • М. А. Юровcкая M. V. Lomonosov Moscow State University, Moscow 119899

Abstract

Under the conditions of the Vilsmeier reaction and also when boiled in biphenyl aminocrotonates, obtained from 2,3,5-trimethyl- and 1,2,3,5-tetramethyl-6-aminoindoles, are easily converted into the corresponding pyrroloquinolines. Similarly, pyrroloquinolines with structures known to be angular are formed during the thermal cyclization of the products from the reaction of these amines with ethoxymethylenemalonic ester.

How to Cite
Yamashkin, S. A.; Kucherenko, N. Y.; Yurovskaya, M. A. Chem. Heterocycl. Compd. 1997, 33, 59. [Khim. Geterotsikl. Soedin. 1997, 69.]

For this article in the English edition, see DOI https://doi.org/10.1007/BF02290747

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Published

1997-01-25

Issue

No. 1 (1997)

Section

Original Papers