SYNTHESIS OF THE FIRST 13-NITROARYL DERIVATIVES OF 8-ACETONYLBERBERINE
DOI:
https://doi.org/10.1007/2569Keywords:
berberine, nitroarene, nucleophilic aromatic substitutionAbstract
For the first time a method for the synthesis of 8-acetonylberberine 13-nitroaryl derivatives has been developed comprising a one-pot reaction of berberine, acetone, and neutral aromatic electrophiles (picryl chloride, 4-chloro-7-nitrobenzofurazan, 4-chloro-5,7-dinitrobenzofurazan). It was found that the reaction of 8-acetonylberberine with these chloronitroarenes does not lead to the formation of the target compounds.
How to Cite
Burov, O. N.; Kurbatov, S. V.; Morozov, P. G.; Kletskii, M. E.; Tatarov, A. V. Chem. Heterocycl. Compd. 2015, 51, 772. [Khim. Geterotsikl. Soedin. 2015, 51, 772.]
For this article in the English edition see DOI 10.1007/s10593-015-1774-6
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Published
2015-09-08
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Letters to the Editor