SYNTHESIS OF SUBSTITUTED 2,5-DIAZABICYCLO[2.2.1]HEPTANES
DOI:
https://doi.org/10.1007/179Keywords:
diazabicycloheptanes, pyrrolidine derivativesAbstract
A new method is proposed for the synthesis of substituted 2,5-diazabicyclo[2.2.1]heptanes from 1-(tert-butoxycarbonyl)-4-tosyloxy-2-(tosyloxymethyl)pyrrolidine. 1H NMR spectroscopy indicated multiple conformations of 2-(tert-butoxycarbonyl)-2,5-diazabicyclo[2.2.1]heptanes in solution.
Authors: M. E. Yakovlev, P. S. Lobanov, and A. A. Potekhin.
English Translation in Chemistry of Heterocyclic Compounds, 2000, 36 (4), pp 429-431