ONE-POT SYNTHESIS OF 3-(2-CYANOPHENYL)-QUINAZOLIN-4(3H)-ONE

Authors

  • W. Szczepankiewicz Institute of Organic Chemistry and Technology, Silesian Technical University
  • J. Suwiński Institute of Organic Chemistry and Technology, Silesian Technical University

DOI:

https://doi.org/10.1007/263

Keywords:

anthranilonitrile, 3-(2-cyanophenyl)quinazolin-4(3H)-one, N-formy-lation

Abstract

Anthranilonitrile reacting with formic acid at room temperature for three days gave 64 % of 3-(2-cyanophenyl)quinazolin-4(3H)-one. Under similar conditions anthranilic acid, 4-nitroaniline and 2,5-dichloroaniline were N-formylated in good yields.

Also published in Chemistry of Heterocyclic Compounds, 2000, 36 (7), pp 809-810

http://link.springer.com/article/10.1007/BF02256914

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Published

2013-02-06

Issue

No. 7 (2000)

Section

Original Papers